Search results for "ACID HYDROLYSIS"

showing 10 items of 38 documents

Structure of a polysaccharide from the lipopolysaccharide of Vibrio vulnificus CECT4602 containing 2-acetamido-2,3,6-trideoxy-3-[(S)- and (R)-3-hydro…

2008

A polysaccharide was isolated by GPC after mild acid treatment of the lipopolysaccharide of Vibrio vulnificus CECT4602 and found to contain L-Rha, D-GlcpNAc and 2-acetamido-2,3,6-trideoxy-3-(3-hydroxybutanoylamino)-L-mannose (L-RhaNAc3NHb). GLC analysis of the trifluoroacetylated (S)-2-octyl esters derived by full acid hydrolysis of the polysaccharide showed that approximately 80% of the 3-hydroxybutanoic acid has the S configuration and approximately 20% the R configuration. The following structure of the polysaccharide was established by (1)H and (13)C NMR spectroscopies, including 2D ROESY and (1)H/(13)C HMBC experiments: [carbohydrate sequence see in text].

Lipopolysaccharideschemistry.chemical_classificationMagnetic Resonance SpectroscopybiologyLipopolysaccharideStereochemistryMolecular Sequence DataPolysaccharides BacterialOrganic ChemistryMannoseGeneral MedicineVibrio vulnificusCarbon-13 NMRbiology.organism_classificationPolysaccharideBiochemistryAnalytical Chemistrychemistry.chemical_compoundCarbohydrate SequencechemistryAcid hydrolysisAcid treatmentMannoseVibrio vulnificusCarbohydrate Research
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A hypotensive procyanidin-glycoside from Rhamnus lycioides ssp. lycioides.

1990

A lyophilized hot water extract of the aerial parts of Rhamnus lycioides L. (Rhamnaceae) produced a lowering of systemic arterial blood pressure in normotensive anaesthetized Wistar rats. An activity-guided fractionation of the methanolic extract led to the isolation of a tetrameric procyanidin-glycoside which produced a clear dose-dependent hypotensive response (1.5-6 mg/kg i.v.). This principle was characterized using acid hydrolysis, thiolytic degradation and spectroscopic methods. It consisted of four flavanol units with a 2,3-cis configuration and with a O-beta-d-glucosylpyranoside function on the epicatechin terminal unit. The interflavan linkage was (4-8).

MaleMagnetic Resonance SpectroscopyStereochemistryBlood PressurePharmacognosyCatechinchemistry.chemical_compoundDrug DiscoveryAnimalsBiflavonoidsProanthocyanidinsGlycosidesRhamnusChromatography High Pressure LiquidPharmacologychemistry.chemical_classificationCarbon IsotopesChromatographyPlants MedicinalbiologyDose-Response Relationship DrugChemistryPlant ExtractsRhamnus lycioidesGlycosideCatechinRats Inbred StrainsPlantsbiology.organism_classificationRatsPlants ToxicRhamnusProanthocyanidinRhamnaceaeAcid hydrolysisHypotensionJournal of ethnopharmacology
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On the Occurrence of Flavonoids in the acrocarpous Mosses

1978

Summary By means of paper chromatography two flavonoids were isolated from the methanolic extract of the moss Mnium undulatum. One substance was identified by chromatographic data, absorption spectra and acid hydrolysis as isovitexin-7-0-glucoside (saponarin). The second substance resists acid hydrolysis and is by chromatography and absorption spectrum identical with apigenin-6,8-di-C-glycoside (viccnin).

chemistry.chemical_compoundPaper chromatographyChromatographyAbsorption spectroscopychemistrySaponarinIsovitexinAcid hydrolysisGeneral MedicineZeitschrift für Pflanzenphysiologie
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Regioselective substitution of 6,7-dichloroquinoline-5,8-dione: synthesis and X-ray crystal structure of 4a,10,11-triazabenzo[3,2-a]fluorene-5,6-dion…

2003

6,7-Dichloroquinoline-5,8-dione (1) was reacted with a number of 2-aminopyridine derivatives. Of the several possible products of this reaction, 4a,10,11-triazabenzo[3,2-a]fluorene-5,6-dione (6), produced by condensation and rearrangement, was obtained as the major product, and its structure was subsequently unambigously determined by X-ray crystallographic study. Ortho-quinones were produced via nucleophilic substitution at position C7, which was unexpected, considering that para-quinones were produced via C6 substitution in the reaction between compound 1 and ethyl acetoacetate in our previous work. Such unexpected nucleophilic substitution at C7 provides an effective, yet simple route, t…

StereochemistryClinical BiochemistryPharmaceutical ScienceAntineoplastic AgentsCrystallography X-RayBiochemistryMedicinal chemistryChemical synthesisInhibitory Concentration 50chemistry.chemical_compoundNucleophilic aromatic substitutionDrug DiscoveryTumor Cells CulturedNucleophilic substitutionHumansMolecular BiologySubstitution reactionFluorenesMolecular StructureOrganic ChemistryQuinonesRegioselectivityStereoisomerismQuinonechemistryDoxorubicinEthyl acetoacetateQuinolinesMolecular MedicineAcid hydrolysisDrug Screening Assays AntitumorBioorganic & Medicinal Chemistry
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Ursane-Type Triterpene Saponins fromZygophyllum geslini

2007

Four new ursane-based triterpene glycosides, compounds 1–4, as well as the known glycosides zygophylosides E, G, and H, and 3-O-(β-D-quinovopyranosyl)quinovic acid 28-(O-β-D-glucopyranosyl) ester, were isolated from the BuOH-soluble fraction of the MeOH/H2O 7 : 3 extracts of Zygophyllum geslini (roots or aerial parts). Their structures were established mainly by 1D- and 2D-NMR techniques, in combination with HR-MS analysis and acid hydrolysis.

chemistry.chemical_classificationbiologyOrganic ChemistryGlycosideFraction (chemistry)Zygophyllumbiology.organism_classificationBiochemistryCatalysisInorganic ChemistryTerpenechemistryTriterpeneDrug DiscoveryOrganic chemistryAcid hydrolysisPhysical and Theoretical ChemistryQuinovic acidHelvetica Chimica Acta
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Nucleophilic substitutions in the isoindole series as a valuable tool to synthesize derivatives with antitumor activity

2011

Abstract A novel synthetic approach to the synthesis of 3-substituted isoindoles through nucleophilic substitution of 3-halo derivatives by charged carbon, and neutral nitrogen, oxygen, and sulfur nucleophiles, assisted by a 1-acyl group, is reported. Aryl-thio-isoindoles, obtained through a direct nucleophilic substitution with sulfur nucleophiles, showed cytotoxic activity, with GI50 values from micromolar to sub-micromolar concentrations, against the total number of cell lines investigated.

chemistry.chemical_classificationKetoneIsoindolesTertiary amineStereochemistryChemistryIsoindoles Nucleophilic substitutionsColchicine analoguesOrganic ChemistryIsoindoles Nucleophilic substitutions; Antitumor activity; Docking; Colchicine analoguesBiochemistryCombinatorial chemistryChemical synthesisSettore CHIM/08 - Chimica FarmaceuticaDockingchemistry.chemical_compoundIsoindoles Nucleophilic substitutionNucleophileColchicine analogueDrug DiscoveryNucleophilic substitutionAcid hydrolysisIsoindoleAntitumor activity
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On the Reaction of 3-Bromo-2-nitrobenzo[b]thiophene 13C-Labeled at C-2 with 3-(Trifluoromethyl)aniline:  A Preliminary Insight into a Nucleophilic Su…

1997

The results of the title reaction have furnished proofs against a rearrangement of the carbon-atom skeleton and for a nitro group shift in the relevant nucleophilic substitution.

Substitution reactionTrifluoromethylStereochemistryKornblum–DeLaMare rearrangementfungiOrganic Chemistrybehavioral disciplines and activitiesbody regionschemistry.chemical_compoundchemistryNucleophilic aromatic substitutionparasitic diseasesNitroNucleophilic substitutionThiopheneAcid hydrolysisThe Journal of Organic Chemistry
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Amino acid profile of milk-based infant formulas

2000

The protein content and amino acid profile of three milk-based infant formulas, two of which were powdered (adapted and follow-on) and the third liquid, were determined to check their compliance with the EU directive and to evaluate whether or not they fulfil an infant's nutritional needs. To obtain the amino acid profile proteins were subjected to acid hydrolysis, prior to which the sulfur-containing amino acids were oxidized with performic acid. The amino acids were derivatized with phenylisothiocyanate (PITC) and then determined by ion-pair reverse phase high performance liquid chromatography (HPLC) In the case of tryptophan a basic hydrolysis was applied and there was no need of derivat…

High-performance liquid chromatographychemistry.chemical_compoundHydrolysisAnimalsHumansmedia_common.cataloged_instanceEuropean UnionAmino AcidsEuropean unionInfant Nutritional Physiological PhenomenaChromatography High Pressure Liquidmedia_commonchemistry.chemical_classificationAnalysis of VariancePerformic acidChromatographyMilk HumanInfant NewbornNutritional RequirementsTryptophanTryptophanInfantLegislation FoodAmino acidMilkchemistryInfant formulaInfant FoodAcid hydrolysisDietary ProteinsFood ScienceInternational Journal of Food Sciences and Nutrition
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A Generalized Synthesis of 3-Amino-5-aryl-, 3-Amino-5-polyfluorophenyl-, and 3-Amino-5-alkyl-1,2,4-oxadiazoles through Ring-degenerate Rearrangements

2002

A generalized synthesis of 3-amino-5-aryl-, 3-amino-5-poly- fluorophenyl- and 3-amino-5-alkyl-1,2,4-oxadiazoles has been developed starting from the 3-amino-5-methyl-1,2,4-oxadiazole as a common synthon. Aroylation or alkanoylation of this aminooxadiazole, followed by thermally- induced ring-degenerate equilibration of resulting 3-acylamino compounds, and final acid hydrolysis of the 3-acetylamino-5-aryl- (or 5-polyfluorophenyl-), or 3- acetylamino-5-alkyl-1,2,4-oxadiazoles counterpart which is formed, gave the expected 3-amino-5-substituted 1,2,4-oxadiazoles. In the case of some 3- aroylamino compounds, yields of final 3-amino-5-aryloxadiazoles are higher than that expected on the basis of…

Pharmacologychemistry.chemical_classificationChemistryArylOrganic ChemistryDegenerate energy levelsSynthonComposition (combinatorics)Ring (chemistry)Medicinal chemistryAnalytical Chemistrychemistry.chemical_compoundAcid hydrolysisAlkylHETEROCYCLES
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Directed Assembly of Cellulose Nanocrystals in Their Native Solid-State Template of a Processed Fiber Cell Wall

2021

Funding Information: I.S. thanks The Academy of Finland (grant no. 300364) for funding this work. C.D. acknowledges funding from FAPESP (grant 13/07932‐6). P.A.P. thanks the Emil Aaltonen Foundation and Academy of Finland (grant no. 315768) for funding and ESRF for beamtime at beamline D2am (experiment 02‐01‐885). Rita Hatakka is acknowledged for her assistance with the GPC measurements. Work of M.L. was supported by the Jane and Aatos Erkko Foundation. The work is a part of the FinnCERES Bioeconomy ecosystem. Publisher Copyright: © 2021 The Authors. Macromolecular Rapid Communications published by Wiley-VCH GmbH Copyright: Copyright 2021 Elsevier B.V., All rights reserved. Nanoparticle ass…

bio-based materialsMaterials scienceporosityPolymers and Plasticsselluloosananoparticle assemblyNanoparticlebio‐based materials02 engineering and technology010402 general chemistry01 natural scienceshuokoisuuschemistry.chemical_compoundHydrolysissymbols.namesakeAdsorptionnanorakenteetCell Wallacid hydrolysisMaterials ChemistryFiberCotton FiberCelluloseCelluloseHydrolysisOrganic Chemistry021001 nanoscience & nanotechnologycellulose0104 chemical scienceschemistryFiber cellChemical engineeringsymbolsNanoparticlesnanohiukkasetnanoselluloosaAcid hydrolysisvan der Waals force0210 nano-technology
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